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                                  350vip浦京集团
                                  师资力量

                                  冯小明     教 授 (中科院院士、博导)

                                  研究方向:不对称合成

                                  联系方式:86-28-8541 8249          Email:xmfeng@scu.edu.cn

                                  个人主页:点击进入

                                  简历:

                                  1981-1988兰州大学化学系有机化学专业学习,获理学学士学位和理学硕士学位。

                                  1993-1996中国科学院化学研究所学习,获理学博士学位。

                                  1988-1993西南师范大学化学系从事有机化学教学和科研工作,历任助教和副教授。

                                  1996-2000中国科学院成都有机化学研究所从事不对称催化反应研究,历任副研究员和研究员,不对称合成联合开放实验室副主任,于1999年被评聘为博士生导师。

                                  1998-1999美国Colorado State University化学系做博士后研究。

                                  2000-至今350vip浦京集团教授,博士生导师。

                                  2002年获国家杰出青年科学基金资助,四川省有突出贡献优秀专家称号;2004年入选四川省学术与技术带头人和获国务院政府特殊津贴;2005年入选教育部重要人才计划特聘教授;2007年获宝钢优秀教师奖,人事部“新世纪百千万人才工程”国家级人选;2008年获教育部“重要人才计划和创新团队发展计划”创新团队资助(学术带头人);2010年获国家创新研究群体资助(学术带头人);2013年当选中国科学院院士;2014年当选英国皇家化学会会士;2020年当选中国化学会创始会士。

                                  ChemistryAn Asian Journal、《有机化学》、《无机化学学报》编委,Angewandte ChemieAdvanced Synthesis & CatalysisCurrent Organic SynthesisAsian Journal of Organic ChemistrySynthesisSynlettChinese Chemical Letters、《应用化学》和《结构化学》顾问编委。

                                  主要研究方向

                                  主要从事新型手性催化剂的设计合成、不对称催化反应、手性药物和生理活性化合物的高效高选择性合成研究。详见课题组主页http://www.scu.edu.cn/chem_asl

                                  主要工作业绩

                                  针对不对称合成中发展新型优势手性催化剂、新反应和新策略等核心问题,进行系统深入的研究。以廉价易得的氨基酸为原料,设计合成了多种具有原创性和特色的优势手性催化剂和配体,其中手性双氮氧化合物被称为“冯氏配体”面向全世界销售,实现了60多类重要不对称反应,如第一例不对称催化α-取代重氮酯与醛的反应,被国外人名反应专著冠名为Roskamp-Feng反应,为一些重要生物活性手性化合物的合成提供有效方法。现已在Acc. Chem. Res., Chem. Rev., J. Am. Chem. Soc., Angew. Chem. Int. Ed., Nat. Commun., CCS Chem.等刊物上发表SCI论文500多篇。研究成果入选了“2011年中国高等学校十大科技进展”,中科院2012《科学发展报告》和《国家自然科学基金资助项目优秀成果选编》。

                                  主要奖励和荣誉 

                                  2009年获教育部高等学校科学研究优秀成果奖自然科学一等奖(第一完成人);2010年获国家自然科学基金委创新研究群体资助(学术带头人);2010年获药明康德“生命化学奖”二等奖;2011年获“中国高等学校十大科技进展”,获中国化学会有机化学委员会颁发的“有机合成创造奖”、获全国优秀博士学位论文指导教师荣誉称号;2012年获国家自然科学奖二等奖(第一完成人);2013年当选中国科学院院士;2014年当选英国皇家化学会会士;2015年获四川大学基础研究年度卓越奖一等奖;2016年获中国化学会“手性化学奖”,四川大学-东土学术创新奖一等奖;2018年获未来科学大奖物质科学奖,中国化学会黄耀曾金属有机化学奖;2019年获教育部高等学校科学研究优秀成果奖自然科学一等奖(第一完成人),何梁何利基金科学与技术进步奖,四川杰出人才奖;2020年获全国创新争先奖章,陈嘉庚科学奖,杰出教学奖,四川省科技杰出贡献奖,2021年入选全国杰出专业技术人才,获中国化学会-中国石油化工股份有限公司化学贡献奖。

                                  代表性成果 (获奖成果、专著、论文、专利)

                                  1.Dong Zhang,# Maoping Pu,# Zhenzhong Liu, Yuqiao Zhou, Zhendong Yang, Xiaohua Liu,* Yun-Dong Wu,* Xiaoming Feng,*Enantioselectiveanti-Dihalogenation of Electron-Deficient Olefin: A Triplet Halo-Radical Pylon Intermediate, J. Am. Chem. Soc.2023,145, 4808−4818.

                                  2.Jinxiu Xu, Yanji Song, Jia Yang, Bingqian Yang, Zhishan Su, Lili Lin,* Xiaoming Feng,* Sterically Hindered and Deconjugative α-Regioselective Asymmetric Mannich Reaction of Meinwald Rearrangement-Intermediate, Angew. Chem. Int. Ed. 2023,62, e202217887.

                                  3.Tangyu Zhan, Liangkun Yang, Qiyou Chen, Rui Weng, Xiaohua Liu,* Xiaoming Feng,* Chiral Lewis Acid-Catalyzed Norrish Type II Cyclization to Synthesize α-Oxazolidinones via Enantioselective Protonation,CCS Chem.2023,5, accepted, DOI: 10.31635/ccschem.022.202202405.

                                  4.Zhikun Wu,# Xiying Zhang,# Nian Xu, Xiaohua Liu,* Xiaoming Feng,* Asymmetric Catalytic Aerobic Oxidative Radical Addition/Hydroxylation/1,4-Aryl Migration Reaction of Olefins, ACS Catal.2023,13, 815−823.

                                  5.Yuhao Mo, Qiyou Chen, Jinzhao Li, Dong Ye, Yuqiao Zhou, Shunxi Dong, Xiaohua Liu,* Xiaoming Feng,* Asymmetric Catalytic Conjugate Addition of Cyanide to Chromones and β‑Substituted Cyclohexenones, ACS Catal.2023,13, 877−886.

                                  6.Shiyang Li, Cefei Zhang, Guihua Pan, Liangkun Yang, Zhishan Su, Xiaoming Feng, Xiaohua Liu,* Enantioselective Photochemical Carbene Insertion into C−C and C−H Bonds of 1,3-Diketones by a Guanidine-Amide Organocatalyst, ACS Catal.2023,13, 4656−4666.

                                  7.Sijing Wang, Cefei Zhang, Da Li, Yuqiao Zhou, Zhishan Su, Xiaoming Feng, Shunxi Dong,* New Chiral N-Heterocyclic Olefin Bifunctional Organocatalysis in α-Functionalization of β-Ketoesters, Sci. China. Chem,2023,66, 147154.

                                  8.Yongyan Zhang, Jin Wu, Lichao Ning, Qianping Chen, Xiaoming Feng, Xiaohua Liu,* Enantioselective Synthesis of Tetrasubstituted Allenes via Addition/Arylation Tandem Reaction of 2-Activated 1,3-Enynes, Sci. China Chem.2023,66, 526533.

                                  9.Ziwei Zhong, Lichao Ning, Yican Lu, Jiuqi Tan, Lili Lin,* Xiaoming Feng,* Asymmetric Catalytic Alkylation of Vinyl Azides with 3-Bromo Oxindoles: Water-assisted Chemo- and Enantiocontrol, Sci. China Chem.2023,66, 799807.

                                  10.Lili Lin, Yuqiao Zhou, Weidi Cao, Shunxi Dong, Xiaohua Liu, Xiaoming Feng,* Progress in N,N′-Dioxide/metal Complex-catalyzed Asymmetric Reactions of Ylides, Sci. Sin. Chem.2023,53, 246258.

                                  11.Siyuan Wang, Yuqiao Zhou, Wanlong Xiao, Zegong Li, Xiaohua Liu,* Xiaoming Feng,* Asymmetric Synthesis of Complex Tricyclo[3.2.2.0] Nonenes from Racemic Norcaradienes: Kinetic Resolution via Diels–Alder Reaction, Chem. Sci.2023,14, 18441851.

                                  12.Shiyu Wang, Chenhao Zhu, Lichao Ning, Dawei Li, Xiaoming Feng,* Shunxi Dong,* Regioselective C–H Alkylation of Anisoles with Olefins by Cationic Imidazolin-2-iminato Scandium(III) Alkyl Complexes, Chem. Sci.,2023,14, 3132−3139.

                                  13.Shunxi Dong, Xiaohua Liu,* Xiaoming Feng,* Asymmetric Catalytic Rearrangements with α‑Diazocarbonyl Compounds, Acc. Chem. Res.2022,55,415−428.

                                  14.Liuzhen Hou, Yuqiao Zhou, Han Yu, Tangyu Zhan, Weidi Cao,* Xiaoming Feng,* Enantioselective Radical Addition to Ketones through Lewis Acid-Enabled Photoredox Catalysis, J. Am. Chem. Soc.2022,144,22140−22149.

                                  15.Xiaobin Lin,# Maoping Pu,# Xinpeng Sang, Shiyang Li, Xiaohua Liu,* Yun-Dong Wu,* Xiaoming Feng,* Asymmetric Catalytic (2+1) Cycloaddition of Thioketones to Synthesize Tetrasubstituted Thiiranes, Angew. Chem. Int. Ed. 2022,61, e202201151.

                                  16.Qianchi Lin, Sujuan Zheng, Long Chen, Jin Wu, Jinzhao Li, Peizhi Liu, Shunxi Dong,* Xiaohua Liu, Qian Peng,* Xiaoming Feng,* Catalytic Regio- and Enantioselective Protonation for the Synthesis of Chiral Allenes: Synergistic Effect of the Counterion and Water, Angew. Chem. Int. Ed. 2022,61,e202203650.

                                  17.Hongkai Wang, Yang Xu, Fangqing Zhang, Yangbin Liu,* Xiaoming Feng,* Bimetallic Palladium/Cobalt Catalysis for Enantioselective Allylic C-H Alkylation via a Transient Chiral Nucleophile Strategy, Angew. Chem. Int. Ed. 2022,61, e202115715.

                                  18.Zhenda Tan, Shibo Zhu, Yangbin Liu,* Xiaoming Feng,* Photoinduced Chemo-, Site- and Stereoselective α-C(sp3)−H Functionalization of Sulfides, Angew. Chem. Int. Ed. 2022,61,e202203374.

                                  19.Wei Wang, Fangqing Zhang, Yangbin Liu,* Xiaoming Feng,* Diastereo- and Enantioselective Construction of Vicinal All-Carbon Quaternary Stereocenters via Iridium/Europium Bimetallic Catalysis, Angew. Chem. Int. Ed. 2022,61, e202208837.

                                  20.Wanlong Xiao, Lichao Ning, Shuang Xin, Shunxi Dong, Xiaohua Liu,* Xiaoming Feng,* Enantioselective [2+2] Cycloaddition of Allenyl Imidewith Mono-, or Disubstituted Alkenes, Angew. Chem. Int. Ed. 2022,61, e202211596.

                                  21.Lifeng Wang, Yuqiao Zhou, Zhishan Su, Fengcai Zhang, Weidi Cao, Xiaohua Liu,* Xiaoming Feng,* [3,3]-Sigmatropic Rearrangements of Naphthyl 1-Propargyl Ethers: para-Propargylation and Catalytic Asymmetric Dearomatization, Angew. Chem. Int. Ed. 2022,61, e202211785.

                                  22.Yang Xu, Hongkai Wang, Zhuang Yang, Yuqiao Zhou, Yangbin Liu,* Xiaoming Feng,* Stereodivergent Total Synthesis of Rocaglaol Initiated by Synergistic Dual-metal-catalyzed Asymmetric Allylation of Benzofuran-3(2H)-one, Chem,2022,8,2011−2022.

                                  23.Yun Liu, Yushuang Chen, Aying Yihuo, Yuqiao Zhou, Xiaohua Liu, Lili Lin,* Xiaoming Feng,* Diastereodivergent Synthesis of Chiral α‑Aminoketones via a Catalytic O−H Insertion/Barnes−Claisen Rearrangement Reaction, ACS Catal.2022,12, 1784−1790.

                                  24.Han Yu, Tangyu Zhan, Yuqiao Zhou, Long Chen, Xiaohua Liu*, Xiaoming Feng,* Visible-Light-Activated Asymmetric Addition of Hydrocarbons to Pyridine-Based Ketones, ACS Catal.2022,12, 5136−5144.

                                  25.Yao Luo, Qi Wei, Liangkun Yang, Yuqiao Zhou, Weidi Cao, Zhishan Su, Xiaohua Liu,* Xiaoming Feng,* Enantioselective Radical Hydroacylation of α,β-Unsaturated Carbonyl Compounds with Aldehydes by Triplet Excited Anthraquinone, ACS Catal.2022,12, 12984−12992.

                                  26.Yan Wang, Aying Yihuo, Lifeng Wang, Shunxi Dong,* Xiaoming Feng,* Catalytic Asymmetric Synthesis of Chiral Azo Compounds via Interrupted Japp–Klingemann Reaction with Aryldiazonium Salts, Sci. China Chem.2022,65, 546−553.

                                  27.Jiawen Lang, Siyuan Wang, Changli He, Xiaohua Liu,* Xiaoming Feng,* Asymmetric Synthesis of Isochromanone Derivatives via Trapping Carboxylic Oxonium Ylides and Aldol Cascade, Chem. Sci.2022,13, 1163−1168.

                                  28.Fangqing Zhang, Bing-Tao Ren, Yuqiao Zhou, Yangbin Liu,* Xiaoming Feng,* Enantioselective Construction of cis-Hydroindole Scaffolds via an Asymmetric Inverse-Electron-Demand Diels–Alder reaction: Application to the Formal Total Synthesis of (+)-Minovincine, Chem. Sci.2022,13, 5562–5567.

                                  29.Liangkun Yang, Wang-Yuren Li, Liuzhen Hou, Tangyu Zhan, Weidi Cao,* Xiaohua Liu, Xiaoming Feng,* Nickel-Catalyzed Asymmetric Photoenolization/Mannich Reaction of (2-Alkylphenyl) Ketones, Chem. Sci.2022,13, 8576–8582.

                                  30.Yi Li, Shuang Xin, Rui Weng, Xiaohua Liu,* Xiaoming Feng,* Asymmetric Synthesis of Chromanone Lactones via Vinylogous Conjugate Addition of Butenolide to 2-Ester Chromones, Chem. Sci.2022,13, 8871–8875.

                                  31.Yangbin Liu, Xiaohua Liu, Xiaoming Feng,* Recent Advances in Metal-catalysed Asymmetric Sigmatropic Rearrangements, Chem. Sci.2022,13, 12290−12308.

                                  32.Fei Tan,#Maoping Pu,# Jun He, Jinzhao Li, Jian Yang, Shunxi Dong, Xiaohua Liu,* Yun-Dong Wu,* Xiaoming Feng,* Catalytic Asymmetric Homologation of Ketones with α-Alkyl-α-diazoesters, J. Am. Chem. Soc.2021,143, 2394−2402.

                                  33.Wei Yang,# Maoping Pu,# Xiaobin Lin, Min Chen, Yanji Song, Xiaohua Liu,* Yun-Dong Wu,* Xiaoming Feng,* Enantioselective Formal Vinylogous N−H Insertion of Secondary Aliphatic Amines Catalyzed by a High-Spin Cobalt(II) Complex, J. Am. Chem. Soc.2021,143, 9648−9656.

                                  34.Wen Liu,# Maoping Pu,# Jun He, Tinghui Zhang, Shunxi Dong, Xiaohua Liu,* Yun-Dong Wu,* Xiaoming Feng,* Iron-Catalyzed Enantioselective Radical Carboazidation and Diazidation of a,b-Unsaturated Carbonyl Compounds, J. Am. Chem. Soc.2021,143,11856−11863.

                                  35.Long Chen,# Maoping Pu,# Shiyang Li, Xinpeng Sang, Xiaohua Liu,* Yun-Dong Wu,* and Xiaoming Feng,* Enantioselective Synthesis of Nitriles Containing a Quaternary Carbon Center by Michael Reactions of Silyl Ketene Imines with 1‑Acrylpyrazoles, J. Am. Chem. Soc.2021,143, 19091–19098.

                                  36.Yong Xia, Xiaohua Liu,* Xiaoming Feng,* Asymmetric Catalytic Reactions of Donor-Acceptor Cyclopropanes, Angew. Chem. Int. Ed.2021,60, 9192–9204.

                                  37.Jinxiu Xu, Yanji Song, Jun He, Shunxi Dong, Lili Lin, Xiaoming Feng,* Asymmetric Catalytic Vinylogous Addition Reactions Initiated by Meinwald Rearrangement of Vinyl Epoxides, Angew. Chem. Int. Ed.2021,60, 1452114527.

                                  38.Li Dai, Wen Liu, Yuqiao Zhou, Zi Zeng, Xinyue Hu, Weidi Cao,* Xiaoming Feng,* Catalytic Asymmetric Halogenation/Semipinacol Rearrangement of 3-Hydroxyl-3-vinyl Oxindoles: A Stereodivergent Kinetic Resolution Process, Angew. Chem. Int. Ed.2021,60, 2659926603.

                                  39.Xinyue Hu, Xiaoxue Tang, Xiying Zhang, LiLi Lin,* Xiaoming Feng,* Catalytic Asymmetric Nakamura Reaction by Gold(I)/chiral N,Nʹ-dioxide-indium(III) or Nickel(II) Synergistic Catalysis, Nat. Commun.2021,12,30123021.

                                  40.Guihua Pan, Changli He, Min Chen, Qian Xiong, Weidi Cao,* Xiaoming Feng,* Synthesis of Dihydroisoquinoline and Dihydropyridine Derivatives via Asymmetric Dearomative Three-component Reaction, CCS Chem.2021,3,20122020.

                                  41.Wanlong Xiao, Yuhao Mo, Jing Guo, Zhishan Su, Shunxi Dong,* Xiaoming Feng,* Catalytic Enantioselective Synthesis of Macrodiolides and Their Application in Chiral Recognition, Chem. Sci.2021,12, 2940−2947.

                                  42.Xia Zhong, Ziwei Zhong, Zhikun Wu, Zhen Ye, Yuxiang Feng, Shunxi Dong, Xiaohua Liu,* Qian Peng,* Xiaoming Feng,* Chiral Lewis Acid-bonded Picolinaldehyde Enables Enantiodivergent Carbonyl Catalysis in Mannich/Condensation Reaction of Glycine Ester, Chem. Sci.2021,12, 43534360.

                                  43.Chaoran Xu, Jianglin Qiao, Shunxi Dong,* Yuqiao Zhou, Xiaohua Liu, Xiaoming Feng,* Asymmetric Synthesis of Dihydro-1,3-dioxepines by Rh(II)/Sm(III) Relay Catalytic Three-component Tandem [4+3]-Cycloaddition, Chem. Sci.2021,12, 54585463.

                                  44.Mingming Guan, Shiyu Wang, Yao Luo, Weidi Cao,* Xiaohua Liu, Xiaoming Feng,* Catalytic Asymmetric Addition of Thiols to Silyl Glyoxylates for Synthesis of Multi-hetero-atom Substituted Carbon Stereocenter, Chem. Sci.2021,12, 7498−7503.

                                  45.Xia Zhong, Jiuqi Tan, Jianglin Qiao, Yuqiao Zhou, Cidan Lv, Zhishan Su, Shunxi Dong,* Xiaoming Feng,* Asymmetric Catalytic Synthesis of Spirocyclobutyl Oxindoles and Beyond via [2+2] Cycloaddition and Sequential Transformations, Chem. Sci.2021,12, 9991−9997.

                                  46.Dong Zhang, Zhisan Su, Qianwen He, Zhikun Wu, Yuqiao Zhou, Chenjing Pan, Xiaohua Liu,* Xiaoming Feng,* Diversified Transformations of Tetrahydroindolizines to Construct Chiral 3-Arylindolizines and Dicarbofunctionalized 1,5-Diketones, J. Am. Chem. Soc.2020,142, 15975−15985.

                                  47.Xiying Zhang, Wangbin Wu, Weidi Cao, Han Yu, Xi Xu, Xiaohua Liu,* Xiaoming Feng,* Enantioselective Radical-Polar Crossover Reactions of Indanonecarboxamides with Alkenes, Angew. Chem. Int. Ed.2020,59, 4846−4850.

                                  48.Yushuang Chen, Yun Liu, Zhaojing Li, Shunxi Dong,* Xiaohua Liu, Xiaoming Feng,* Tandem Insertion/[1,3]-Rearrangement: Highly Enantioselective Construction of a-Aminoketones,Angew. Chem. Int. Ed.2020,59, 8052−8056.

                                  49.Tengfei Kang, Liuzhen Hou, Sai Ruan, Weidi Cao, Xiaohua Liu,* Xiaoming Feng,* Lewis acid-catalyzed asymmetric reactions of β,γ-unsaturated 2-acyl imidazoles, Nat. Commun.2020,11, 3869.

                                  50.Xiaobin Lin, Zheng Tan, Wenkun Yang, Wei Yang, Xiaohua Liu,* Xiaoming Feng,* Chiral Cobalt(ΙΙ) Complex Catalyzed Asymmetric [2,3]-Sigmatropic Rearrangement of Allylic Selenides with α-Diazo Pyrazoleamides, CCS Chem.2020,2, 1423–1433.

                                  51.Jian Xu, Ziwei Zhong, Mingyi Jiang, Yuqiao Zhou, Xiaohua Liu,* Xiaoming Feng,* Asymmetric Catalytic Concise Synthesis of Hetero-3,3ʹ-Bisoxindoles for the Construction of Bispyrroloindoline Alkaloids, CCS Chem. 2020,2, 1894–1902.

                                  52.Zhen Wang, Xiaohua Liu,* Xiaoming Feng,* Asymmetric Catalysis Enabled by Chiral N,N'-Dioxide–Nickel(II) Complexes, Aldrichimica ACTA,2020,53, 3−10.

                                  53.Qianchi Lin, Bowen Hu, Xi Xu, Shunxi Dong, Xiaohua Liu,* Xiaoming Feng,* Chiral N,Nʹ-Dioxide/Mg(OTf)2 Complex-Catalyzed Asymmetric [2,3]-Rearrangement of in situ Generated Ammonium Salts, Chem. Sci. 2020,11, 3068−3073.

                                  54.Bin Shen, Qianwen He, Shunxi Dong, Xiaohua Liu,* Xiaoming Feng,* Chiral Cobalt(II) Complex Catalyzed Enantioselective Aza-Piancatelli Rearrangement/Diels-Alder Cascade Reaction, Chem. Sci. 2020,11, 3862−3867.

                                  55.Lifeng Wang, Pengfei Zhou,  Qianchi Lin,  Shunxi Dong,  Xiaohua Liu,* Xiaoming Feng,* Chiral Fe(II) Complex Catalyzed Enantioselective [1,3] O-to-C Rearrangement of Alkyl Vinyl Ethers and Synthesis of Chromanols and Beyond, Chem. Sci. 2020,11,10101-10106.

                                  56.Ziwei Zhong, Zhijie Xiao, Xiaohua Liu, Weidi Cao,* Xiaoming Feng,*Catalytic Asymmetric Synthesis of 3,2'-Pyrrolinyl Spirooxindoles via Conjugate Addition/Schmidt-type Rearrangement of Vinyl Azides and (E)-Alkenyloxindoles,Chem. Sci. 2020,11,11492-11497.

                                  57.Bin Shen, Qianwen He, Shunxi Dong, Xiaohua Liu,* Xiaoming Feng,* Chiral Cobalt(II) Complex Catalyzed Enantioselective Aza-Piancatelli Rearrangement/Diels-Alder Cascade Reaction, Chem. Sci. 2020,11, 3862−3867.

                                  58.Weidi Cao, Xiaohua Liu, Xiaoming Feng,* ChiralN,Nʹ-dioxide and Their Metal Complexes in Asymmetric Catalysis (in Chinese), Chin. Sci. Bull.2020,65, 2941−2951.

                                  59.Qian Xiong, Shunxi Dong, Yushuang Chen, Xiaohua Liu,* Xiaoming Feng,* Asymmetric Synthesis of Tetrazole and Dihydroisoquinoline Derivatives by Isocyanidebased Multicomponent Reactions, Nat. Commun.2019,10, 2116.

                                  60.Tengfei Kang, Weidi Cao, Liuzhen Hou, Qiong Tang, Sijia Zou, Xiaohua Liu, Xiaoming Feng,* Chiral Zinc(II)-Catalyzed Enantioselective Tandem a-Alkenyl Addition/Proton Shift Reaction of Silyl Enol Ethers with Ketimines, Angew. Chem. Int. Ed.2019,58, 2464–2468.

                                  61.Shulin Ge, Weidi Cao, Tengfei Kang, Bowen Hu, Hang Zhang, Zhishan Su, Xiaohua Liu, Xiaoming Feng,* Bimetallic Catalytic Asymmetric Tandem Reaction of β-Alkynyl Ketones to Synthesize 6,6-Spiroketals, Angew. Chem. Int. Ed.2019,58,4017–4021.

                                  62.Haifeng Zheng, Yan Wang, Chaoran Xu, Qian Xiong, Lili Lin, Xiaoming Feng,* Diversified 1,6-Enynes Cycloisomerization/Diels-Alder Reactions via Bimetallic Relay Asymmetric Catalysis, Angew. Chem. Int. Ed.2019,58, 5327–5331.

                                  63.Qiong Tang, Kai Fu, Peiran Ruan, Shunxi Dong,* Zhishan Su, Xiaohua Liu, Xiaoming Feng,* Asymmetric Catalytic Formal 1,4-Allylation of b,g-Unsaturateda-Ketoesters: Allylboration/Oxy-Cope Rearrangement, Angew. Chem. Int. Ed.2019,58, 11846–11851.

                                  64.Xiaobin Lin, Wei Yang, Wenkun Yang, Xiaohua Liu,* and Xiaoming Feng,* Asymmetric Catalytic [2,3] Stevens and Sommelet–Hauser Rearrangements of a-Diazo Pyrazoleamides with Sulfides, Angew. Chem. Int. Ed.2019,58, 13492–13498.

                                  65.Chaoran Xu, Kaixuan Wang, Dawei Li, Lili Lin,* and Xiaoming Feng,* Asymmetric Synthesis of Oxa-Bridged Oxazocines by Rh(II)/Zn(II) Relay Catalytic [4+3] Cycloaddition Reaction, Angew. Chem. Int. Ed.2019,58, 18438–18442.

                                  66.Yu Zhang, Fengcai Zhang, Long Chen, Jian Xu, Xiaohua Liu,* Xiaoming Feng,* Asymmetric Synthesis of P-Stereogenic Compounds via Thulium(III)-Catalyzed Desymmetrization of Dialkynylphosphine Oxides, ACS Catal.2019,9, 4834−4840.

                                  67.Wangbin Wu, Weidi Cao, Linfeng Hu, Zhishan Su, Xiaohua Liu,* and Xiaoming Feng,* Asymmetric Baeyer–Villiger Oxidation: Classical and Parallel Kinetic Resolution of 3-Substituted Cyclohexanones and Desymmetrization of meso-Disubstituted Cycloketones, Chem. Sci.2019,10, 7003−7008.

                                  68.Ke Zheng, Xiaohua Liu, Xiaoming Feng,* Recent Advances in Metal-Catalyzed Asymmetric 1,4-Conjugate Addition (ACA) of Nonorganometallic Nucleophiles, Chem. Rev. 2018,118, 75867656.

                                  69.Xiaobin Lin, Yu Tang, Wei Yang, Fei Tan, Lili Lin, Xiaohua Liu,* Xiaoming Feng,* Chiral Nickel(II) Complex Catalyzed Enantioselective Doyle-Kirmse Reaction of α-Diazo Pyrazoleamides, J. Am. Chem. Soc.2018,140, 3299–3305.

                                  70.Haifeng Zheng, Yan Wang, Chaoran Xu, Xi Xu, Lili Lin, Xiaohua Liu,* Xiaoming Feng,* Stereodivergent Synthesis of Vicinal Quaternary-quaternary Stereocenters and Bioactive Hyperolactones, Nat. Commun. 2018, 1968−1974.

                                  71.Xi Xu, Jianlin Zhang, Shunxi Dong, Lili Lin, Xiaobin Lin, Xiaohua Liu, Xiaoming Feng,* Nickel(II)-Catalyzed Asymmetric Propargyl [2,3] Wittig Rearrangement of Oxindole Derivatives: A Chiral Amplification Effect, Angew. Chem. Int. Ed.2018,57, 8734–8738.

                                  72.Yuhang Zhou, Lili Lin, Xiaohua Liu,* Xinyue Hu, Yan Lu, Xiying Zhang, Xiaoming Feng,* Catalytic Asymmetric Diels-Alder Reaction/[3,3] Sigmatropic Rearrangement Cascade of 1-Thiocyanatobutadienes,Angew. Chem. Int. Ed.2018,57, 9113–9116.

                                  73.Dong Zhang, Lili Lin, Jian Yang, Xiaohua Liu, Xiaoming Feng,* Asymmetric Synthesis of Tetrahydroindolizines by Bimetallic Relay Catalyzed Cycloaddition of Pyridinium Ylides, Angew. Chem. Int. Ed.2018,57, 12323–12327.

                                  74.Fei Tan, Xiaohua Liu,* Yan Wang, Shunxi Dong, Han Yu, Xiaoming Feng,* Chiral Lewis Acid Catalyzed Reactions of a-Diazoester Derivatives: Construction of Dimeric Polycyclic Compounds, Angew. Chem. Int. Ed.2018,57, 16176–16179.

                                  75.Yushuang Chen, Shunxi Dong, Xi Xu, Xiaohua Liu, Xiaoming Feng,* Bimetallic Rhodium(II)/Indium(III) Relay Catalysis for Tandem Insertion/Asymmetric Claisen Rearrangement, Angew. Chem. Int. Ed.2018,57, 16554–16558.

                                  76.Xiaohua Liu, Xiaoming Feng,* Dual Nickel and Br➢nsted Acid Catalysis for Hydroalkenylation, Angew. Chem. Int. Ed.2018,57, 16604–16605

                                  77.Yali Xu, Fenzhen Chang, Weidi Cao, Xiaohua Liu, Xiaoming Feng,* Catalytic Asymmetric Chemodivergent C2 Alkylation and [3 + 2]-Cycloaddition of 3‑Methylindoles with Aziridines,ACS Catal.2018,8, 10261–10266.

                                  78.Yulong Kuang, Bin Shen, Li Dai, Qian Yao, Xiaohua Liu,* Lili Lin, Xiaoming Feng,* Diastereodivergent Asymmetric Michael-Alkylationreactions Using Chiral N,N′-Dioxide/Metal Complexes, Chem. Sci.2018,9, 688–692.

                                  79.Xiaohua Liu, Shunxi Dong, Lili Lin, Xiaoming Feng,* Chiral Amino Acids-Derived Catalysts and Ligands, Chin. J. Chem.2018,36, 791–797.

                                  80.Xiaohua Liu, Haifeng Zheng, Yong Xia, Lili Lin, Xiaoming Feng,* Asymmetric Cycloaddition and Cyclization Reactions Catalyzed by ChiralN,N′‑Dioxide-Metal Complexes, Acc. Chem. Res.2017,50, 2621-2631.

                                  81.Pengfei Zhou, Lili Lin, Long Chen, Xia Zhong, Xiaohua Liu, Xiaoming Feng,* Iron-Catalyzed Asymmetric Haloazidation of α,β-Unsaturated Ketones: Construction of Organic Azides with Two Vicinal Stereocenters, J. Am. Chem. Soc.2017,139, 13414-13419.

                                  82.Jianfeng Zheng, Lili Lin, Li Dai, Qiong Tang, Xiaohua Liu,* Xiaoming Feng,* Nickel-Catalyzed Conjugate Addition of Silyl Ketene Imines to In Situ Generated Indol-2-ones: Highly Enantioselective Construction of Vicinal All-Carbon Quaternary Stereocenters, Angew. Chem. Int. Ed.2017,56, 13107-13111.

                                  83.Jun Li, Lili Lin, Bowen Hu, Pengfei Zhou, Tianyu Huang, Xiaohua Liu,* Xiaoming Feng,* Gold(I)/Chiral N,N’-Dioxide–Nickel(II) Relay Catalysis for Asymmetric Tandem Intermolecular Hydroalkoxylation/Claisen Rearrangement, Angew. Chem. Int. Ed.2017,56, 885-888.

                                  84.Tianyu Huang, Xiaohua Liu,* Jiawen Lang, Jian Xu, Lili Lin, Xiaoming Feng,* Asymmetric Aerobic Oxidative Cross-Coupling of Tetrahydroisoquinolines with Alkynes, ACS Catal.2017,7, 5654-5660.

                                  85.Jie Ji, Lili Lin, Qiong Tang, Tengfei Kang, Xiaohua Liu, Xiaoming Feng,* Highly Efficient Asymmetric Synthesis of Chiral γ‑Alkenyl Butenolides Catalyzed by Chiral N,N′‑Dioxide-Scandium(III) Complexes, ACS Catal.2017,7, 3763-3767.

                                  86.Yuting Liao, Baixin Zhou, Yong Xia, Xiaohua Liu,* Lili Lin, Xiaoming Feng,* Asymmetric [3 + 2] Cycloaddition of 2,2′-Diester Aziridines To Synthesize Pyrrolidine Derivatives, ACS Catal.2017,7, 3934-3939.

                                  87.Xiangjin Lian, Lili Lin, Kai Fu, Baiwei Ma, Xiaohua Liu, Xiaoming Feng,* A new approach to the asymmetric Mannich reaction catalyzed by chiral N,N’-dioxide-metal complexes, Chem. Sci.,2017,8, 1238-1242.

                                  88.Yu Zhang, Yuting Liao, Xiaohua Liu,*Xi Xu, Lili Lin, Xiaoming Feng,* Catalytic asymmetric hydroxylative dearomatization of 2-naphthols: synthesis of lacinilene derivatives, Chem. Sci.2017,8, 6645-6649.

                                  89.Yong Xia, Lili Lin, Fenzhen Chang, Yuting Liao, Xiaohua Liu,* and Xiaoming Feng,* Asymmetric Ring Opening/Cyclization/Retro-Mannich Reaction of Cyclopropyl Ketones with Aryl 1,2-Diamines for the Synthesis of Benzimidazole Derivatives, Angew. Chem. Int. Ed.2016,55, 12228-12232.

                                  90.Haipeng Hu, Yangbin Liu, Lili Lin, Yuheng Zhang, Xiaohua Liu,* and Xiaoming Feng,* Kinetic Resolution of 2H-Azirines by Asymmetric Imine Amidation, Angew. Chem. Int. Ed.2016,55, 10098-10101.

                                  91.Qian Yao, Yuting Liao, Lili Lin, Xiaobin Lin, Jie Ji, Xiaohua Liu,* and Xiaoming Feng,* Efficient Synthesis of Chiral Trisubstituted 1,2-Allenyl Ketones by Catalytic Asymmetric Conjugate Addition of Malonic Esters to Enynes, Angew. Chem. Int. Ed.2016,55, 1859-1863.

                                  92.Yangbin Liu, Xiaohua Liu,* Haipeng Hu, Jing Guo, Yong Xia, Lili Lin, and Xiaoming Feng,* Synergistic Kinetic Resolution and Asymmetric Propargyl Claisen Rearrangement for the Synthesis of Chiral Allenes, Angew. Chem. Int. Ed.2016,55, 4054-4058.

                                  93.Tengfei Kang, Shulin Ge, Lili Lin, Yan Lu, Xiaohua Liu,* and Xiaoming Feng,* A Chiral N,N′-Dioxide–ZnII Complex Catalyzes the Enantioselective [2+2] Cycloaddition of Alkynones with Cyclic Enol Silyl Ethers, Angew. Chem. Int. Ed.2016,55, 5541-5544.

                                  94.Jun Li, Lili Lin, Bowen Hu, Xiangjin Lian, Gang Wang, Xiaohua Liu,* and Xiaoming Feng,* Bimetallic Gold(I)/Chiral N,N′-Dioxide Nickel(II) Asymmetric Relay Catalysis: Chemo- and Enantioselective Synthesis of Spiroketals and Spiroaminals, Angew. Chem. Int. Ed.2016,55, 6075-6078.

                                  95.Pengfei Zhou, Yunfei Cai, Xia Zhong, Weiwei Luo, Tengfei Kang, Jun Li, Xiaohua Liu,* Lili Lin, and Xiaoming Feng,* Catalytic Asymmetric Intra- and Intermolecular Haloetherification of Enones: An Efficient Approach to (-)-Centrolobine, ACS Catal.2016,6, 7778-7783.

                                  96.Gang Wang, Xiaohua Liu,*, Yushuang Chen, Jian Yang, Jun Li, Lili Lin, and Xiaoming Feng,* Diastereoselective and Enantioselective Alleno-aldol Reaction of Allenoates with Isatins to Synthesis of Carbinol Allenoates Catalyzed by Gold, ACS Catal.2016,6, 2482-2486.

                                  97.Yali Xu, Yuting Liao, Lili Lin, Yuhang Zhou, Jun Li, Xiaohua Liu, and Xiaoming Feng,* Catalytic Asymmetric Inverse-Electron Demand 1,3-Dipolar Cycloaddition of Isoquinolinium Methylides with Enecarbamates by a Chiral N,N′-Dioxide/Ag(I) Complex, ACS Catal.2016,6, 589-592.

                                  98.Jing Guo, Yangbin Liu, Xiangqiang Li, Xiaohua Liu,* Lili Lin and Xiaoming Feng,* Nickel(II)-catalyzed enantioselective cyclopropanation of 3-alkenyl-oxindoles with phenyliodonium ylide via free carbine, Chem. Sci.2016,7, 2717-2721.

                                  99.Yuting Liao, Xiaohua Liu,* Yu Zhang, Yali Xu, Yong Xia, Lili Lin and Xiaoming Feng,* Asymmetric [3 + 2] cycloaddition of donor–acceptor aziridines with aldehydes via carbon–carbon bond cleavage, Chem. Sci.2016,7, 3775-3779.

                                  100.Weiwei Luo, Xiao Yuan, Lili Lin, Pengfei Zhou, Xiaohua Liu* and Xiaoming Feng,* A N,N′-dioxide/Mg(OTf)2 complex catalyzed enantioselective a-addition of isocyanides to alkylidene malonates, Chem. Sci.2016,7, 4736-4740.

                                  101.Yong Xia, Xiaohua Liu*, Haifeng Zheng, Lili Lin, Xiaoming Feng,* A symmetric Synthesis of 2,3-Dihydropyrroles by Ring-Opening/Cyclization of Cyclopropyl Ketones Using Primary Amines, Angew. Chem. Int. Ed. 2015,54,227-230.

                                  102.Yong Xia, Lili Lin, Fenzhen Chang, Xuan Fu, Xiaohua Liu*, Xiaoming Feng,* Asymmetric Ring-Opening of Cyclopropyl Ketones with Thiol, Alcohol, and Carboxylic Acid Nucleophiles Catalyzed by a Chiral N,N′-Dioxide–Scandium(III) Complex, Angew. Chem. Int. Ed.2015,54,13748-13752.

                                  103.Haifeng Zheng, Xiaohua Liu*, Chaoran Xu, Yong Xia, Lili Lin, Xiaoming Feng,* Regio- and Enantioselective Aza-Diels–Alder Reactions of 3-Vinylindoles: A Concise Synthesis of the Antimalarial Spiroindolone NITD609, Angew.Chem.Int. Ed.2015,54,10958-10962.

                                  104.Jiannan Zhao, Bing Fang, Weiwei Luo, Xiaoyu Hao, Xiaohua Liu, Lili Lin, Xiaoming Feng,* Enantioselective Construction of Vicinal Tetrasubstituted Stereocenters by the Mannich Reaction of Silyl Ketene Imines with Isatin-Derived Ketimines, Angew. Chem. Int. Ed. 2015,54,241-244.

                                  105.Wei Li, Fei Tan, Xiaoyu Hao, Gang Wang, Yu Tang, Xiaohua Liu, Lili Lin, Xiaoming Feng,* Catalytic Asymmetric Intramolecular Homologation of Ketones with α-Diazoesters: Synthesis of Cyclic α-Aryl/Alkyl β-Ketoesters, Angew. Chem. Int. Ed. 2015,54,1608-1611.

                                  106.Xiaohu Zhao, Xiaohua Liu*, Hongjiang Mei, Jing Guo, Lili Lin, Xiaoming Feng,* Asymmetric Dearomatization of Indoles through a Michael/Friedel-Crafts-Type Cascade To Construct Polycyclic Spiroindolines, Angew. Chem. Int. Ed.2015,54,4032-4035.

                                  107.Yin Zhu, Xiaohua Liu,* Shunxi Dong, Yuhang Zhou, Wei Li, Lili Lin, Xiaoming Feng,* Asymmetric NH Insertion of Secondary and Primary Anilines under the Catalysis of Palladium and Chiral Guanidine Derivatives, Angew. Chem. Int. Ed. 2014,53, 1636-1640.

                                  108.Yangbin Liu, Haipeng Hu, Haifeng Zheng, Yong Xia, Xiaohua Liu, Lili Lin, Xiaoming Feng,* Nickel(II)-Catalyzed Asymmetric Propargyl and Allyl Claisen Rearrangements to Allenyl- and Allyl-Substituted β-Ketoesters, Angew. Chem. Int. Ed. 2014,53, 11579-11582.

                                  109.Xiaohua Liu, Lili Lin and Xiaoming Feng,* Chiral N,N′-Dioxide Ligands: Synthesis, Coordination Chemistry and Asymmetric Catalysis, Org. Chem. Front.,2014,1, 298-302.

                                  110.Shunxi Dong, Xiaohua Liu*, Yin Zhu, Peng He, Lili Lin, Xiaoming Feng,* Organocatalytic Oxyamination of Azlactones: Kinetic Resolution of Oxaziridines and Asymmetric Synthesis of Oxazolin-4-ones, J. Am. Chem. Soc.2013,135, 10026-10029.

                                  111.Jiannan Zhao, Xiaohua Liu, Weiwei Luo, Mingsheng Xie, Lili Lin, Xiaoming Feng,* Asymmetric Synthesis of β-Amino Nitriles through a ScIII-Catalyzed Three-Component Mannich Reaction of Silyl Ketene Imines, Angew. Chem. Int. Ed.2013,52, 3473-3477.

                                  112.Mingsheng Xie, Xiaohua Liu, Xiaoxia Wu, Yunfei Cai, Lili Lin, Xiaoming Feng,* Catalytic Asymmetric [8+2] Cycloaddition: Synthesis of Cycloheptatriene-Fused Pyrrole Derivative, Angew. Chem. Int. Ed.2013,52, 5604-5607.

                                  113.Jing Guo, Shunxi Dong, Yulong Zhang, Yulong Kuang, Xiaohua Liu, Lili Lin, Xiaoming Feng,* Chiral Scandium(III)-Catalyzed Enantioselective α-Arylation of N-Unprotected 3-Substituted Oxindoles with Diaryliodonium Salts, Angew. Chem. Int. Ed.2013,52, 10245-10249.

                                  114.Wei Li, Xiaohua Liu, Fei Tan, Xiaoyu Hao, Jianfeng Zheng, Lili Lin, Xiaoming Feng,* Catalytic Homologation of α-Ketoesters with α-Diazoesters: Enantioselective Synthesis of Succinate Derivatives with Chiral Quaternary Centers, Angew. Chem. Int. Ed.2013,52, 10883-10886.

                                  115.Ke Zheng, Xiaohua Liu, Song Qin, Mingsheng Xie, Lili Lin, Changwei Hu, Xiaoming Feng,* Completely OH-Selective FeCl3-Catalyzed Prins Cyclization: Highly Stereoselective Synthesis of 4-OH-Tetrahydropyrans, J. Am. Chem. Soc.2012,134, 17564-17573.

                                  116.Lin Zhou, Xiaohua Liu, Jie Ji, Yuheng Zhang, Lili Lin, Xiaoming Feng,* Enantioselective Baeyer−Villiger Oxidation: Desymmetrization of Meso Cyclic Ketones and Kinetic Resolution of Racemic 2‑Arylcyclohexanones, J. Am. Chem. Soc.2012,134, 17023-17026.

                                  117.Wei Li, Xiaohua Liu, Xiaoyu Hao, Yunfei Cai, Lili Lin, Xiaoming Feng,* ACatalytic Asymmetric Ring-Expansion Reaction of Isatins and α-Alkyl-α-Diazoesters: Highly Efficient Synthesis of Functionalized 2-Quinolone Derivatives, Angew. Chem. Int. Ed.2012,51, 8644-8647.

                                  118.Zhen Wang, Zhenling Chen, Sha Bai, Wei Li, Xiaohua Liu, Lili Lin, Xiaoming Feng,* Highly Z-Selective Asymmetric Conjugate Addition of Alkynones with Pyrazol-5-ones Promoted by N,N′-Dioxide–Metal Complexes, Angew. Chem. Int. Ed. 2012,51, 2776-2779.

                                  119.Ke Shen, Xiaohua Liu, Lili Lin, Xiaoming Feng,* Recent Progress in Enantioselective Synthesis of C3-functionalized Oxindoles: Rare Earth Metals Take Action,Chem. Sci.2012,3, 327-334.

                                  120.Yangyang Chu, Xiaohua Liu, Wei Li, Xiaolei Hu, Lili Lin and Xiaoming Feng,* Asymmetric Catalytic Epoxidation of α,β-Unsaturated Carbonyl Compounds with Hydrogen Peroxide: Additive-free and Wide Substrate Scope, Chem. Sci.2012,3, 1996-2000.

                                  121.Ke Zheng, Lili Lin, Xiaoming Feng,* Chiral N,N′-Dioxide-Ni(II) Complex Catalyzed Asymmetric Carbonyl-Ene Reaction Of Ethyl Trifluoropyruvate, Acta Chim. Sinica 2012,70, 1785-1790.

                                  122.Xiaohua Liu, Lili Lin, Xiaoming Feng,* ChiralN,N′-Dioxides: New Ligands and Organocatalysts for Catalytic Asymmetric Reactions, Acc. Chem. Res.2011,44, 574-587.

                                  123.Jun Wang, Xiaohua Liu, Xiaoming Feng,* Asymmetric Strecker Reactions, Chem. Rev.2011,111, 6947-6983.

                                  124.Wei Li, Xiaohua Liu, Xiaoyu Hao, Xiaolei Hu, Yangyang Chu, Weidi Cao, Song Qin, Changwei Hu, Lili Lin, Xiaoming Feng,* New Electrophilic Addition of α-Diazoesters with Ketones for Enantioselective C-N Bond Formation, J. Am. Chem. Soc.2011,133,15268-15271.

                                  125.Yunfei Cai, Xiaohua Liu, Jun Jiang, Weiliang Chen, Lili Lin, Xiaoming Feng,* Catalytic Asymmetric Chloroamination Reaction of α,β-Unsaturated γ-Keto Esters and Chalcones, J. Am. Chem. Soc.2011,133, 5636-5639.

                                  126.Ke Shen, Xiaohua Liu, Gang Wang, Lili Lin, and Xiaoming Feng,* Facile and Efficient Enantioselective Hydroxyamination Reaction: Synthesis of 3-Hydroxyamino-2-Oxindoles Using Nitrosoarenes, Angew. Chem. Int. Ed.2011,50, 4684-4688.

                                  127.Zhen Wang, Zhigang Yang, Donghui Chen, Xiaohua Liu, Lili Lin, Xiaoming Feng,* Highly Enantioselective Michael Addition of Pyrazolin-5-ones Catalyzed by Chiral N,N′-dioxide-Lanthanide(III) Complex: Metal Directed Reversal of Enantioselectivity, Angew. Chem. Int. Ed.2011,50, 4928-4932.

                                  128.Ke Zheng, Chengkai Yin, Xiaohua Liu, Lili Lin, Xiaoming Feng,* Catalytic Asymmetric Addition of Alkyl Enol Ethers to 1,2-Dicarbonyl Compounds: Highly Enantioselective Synthesis of Substituted 3-Alkyl-3-Hydroxyoxindoles, Angew. Chem. Int. Ed.2011,50, 2573-2577.

                                  129.Yunfei Cai, Xiaohua Liu, Jun Li, Weiliang Chen, Wentao Wang, Lili Lin, Xiaoming Feng,* Asymmetric Iodoamination of Chalcones and 4-Aryl-4-oxobutenoates Catalyzed by a Complex Based on Scandium (III) and aN,N′-Dioxide Ligand, Chem. Eur. J.2011,17, 14916-14921.

                                  130.Wei Li, Jun Wang, Xiaolei Hu, Ke Shen, Wentao Wang, Yangyang Chu, Lili Lin, Xiaohua Liu, Xiaoming Feng,* Catalytic Asymmetric Roskamp Reaction of α-Alkyl-α-diazoesters with Aromatic Aldehydes: Highly Enantioselective Synthesis of α-Alkyl-β-keto Esters, J. Am. Chem. Soc. 2010,132, 8532-8533.

                                  131.Shunxi Dong, Xiaohua Liu, Xiaohong Chen, Fang Mei, Yulong Zhang, Bo Gao, Lili Lin, Xiaoming Feng,* Chiral Bisguanidine-Catalyzed Inverse-Electron-Demand Hetero-Diels−Alder Reaction of Chalcones with Azlactones, J. Am. Chem. Soc. 2010,132, 10650-10651.

                                  132.Yunfei Cai, Xiaohua Liu, Yonghai Hui, Jun Jiang, Wentao Wang, Weiliang Chen, Lili Lin, Xiaoming Feng,* Catalytic Asymmetric Bromoamination of Chalcones: Highly Efficient Synthesis of Chiral α-Bromo-β-Amino Ketone Derivatives,Angew. Chem. Int. Ed.2010,49, 6160-6164.

                                  133.Zongrui Hou, Jun Wang, Peng He, Jing Wang, Bo Qin, Xiaohua Liu, Lili Lin, Xiaoming Feng,* Highly Enantioselective Insertion of Carbenoids into N-H Bonds Catalyzed by Copper(I) Complexes of Rigid BINOL Derivatives, Angew. Chem. Int. Ed.2010,49, 4763-4766.

                                  134.Yonghai Hui, Jun Jiang, Wentao Wang, Weiliang Chen, Yunfei Cai, Lili Lin, Xiaohua Liu, Xiaoming Feng,* Highly Enantioselective Conjugate Addition of Thioglycolate to Enones Using Mild Lanthanum Catalysis: Lower Catalyst Loading and Remarkably Chiral Amplification, Angew. Chem. Int. Ed.2010,49, 4290-4293.

                                  135.Mingsheng Xie, Xiaohong Chen, Yin Zhu, Bo Gao, Lili Lin, Xiaohua Liu, Xiaoming Feng,* Asymmetric Three-Component Inverse Electron-Demand Aza-Diels-Alder Reaction: Efficient Synthesis of Ring-Fused Tetrahydroquinolines, Angew. Chem. Int. Ed.2010,49, 3799-3802.

                                  136.Ke Shen, Xiaohua Liu, Wentao Wang, Gang Wang, Weidi Cao, Wei Li, Xiaolei Hu, Lili Lin, Xiaoming Feng,* Highly Enantioselective Synthesis of 1,3-Bis(hydroxymethyl)-2-oxindoles from Unprotected Oxindoles and Formalin Using a Chiral Nd(III)Complex,Chem. Sci.2010,1, 590-595.

                                  137.Zhipeng Yu, Xiaohua Liu, Lin Zhou, Lili Lin, Xiaoming Feng,* Bifunctional Guanidine via an Amino Amide Skeleton for Asymmetric Michael Reactions of β-Ketoesters with Nitroolefins: A Concise Synthesis of Bicyclic β-Amino Acids, Angew. Chem. Int. Ed.2009,48, 5195-5198.

                                  138.Jun Wang, Wentao Wang, Wei Li, Xiaolei Hu, Ke Shen, Cheng Tan, Xiaohua Liu, Xiaoming Feng,* Asymmetric Cyanation of Aldehydes, Ketones, Aldimines, and Ketimines Catalyzed by a Versatile Catalyst Generated from Cinchona Alkaloid, Achiral Substituted 2,2’-Biphenol and Tetraisopropyl Titanate, Chem. Eur. J.2009,15, 11642-11659.

                                  139.Xiaohua Liu, Lili Lin, Xiaoming Feng,* Amide-Based Bifunctional Organocatalysts in Asymmetric Reactions, Chem. Commun.2009, 6145-6158.

                                  140.Ke Zheng, Jian Shi, Xiaohua Liu, Xiaoming Feng,* Asymmetric Carbonyl-Ene Reaction Catalyzed by Chiral N,N′-Dioxide-Nickel(II) Complex: Remarkably Broad Substrate Scope, J. Am. Chem. Soc.2008,130, 15770-15771.

                                  141.Jie Liu, Zhigang Yang, Zhen Wang, Fei Wang, Xiaohong Chen, Xiaohua Liu, Xiaoming Feng,* Zhishan Su, Changwei Hu*, Asymmetric Direct Aldol Reaction of Functionalized Ketones Catalyzed by Amine Organocatalysts Based on Bispidine, J. Am. Chem. Soc.2008,130, 5654-5655.

                                  142.Lijia Wang, Xiaohua Liu, Zhenhua Dong, Xuan Fu, Xiaoming Feng,* Asymmetric Intramolecular Oxa-Michael Addition of Activated α,β-Unsaturated Ketones Catalyzed by a Chiral N,N′-Dioxide Nickel(II) Complex: Highly Enantioselective Synthesis of Flavanones,Angew. Chem., Int. Ed.2008,47, 8670-8673.

                                  143.Xu Yang, Xin Zhou, Lili Lin, Lu Chang, Xiaohua Liu, Xiaoming Feng,* Highly Enantioselective Direct Michael Addition of Nitroalkanes to Nitroolefins Catalyzed by La(OTf)3/N,N′-Dioxide Complexes,Angew. Chem. Int. Ed.2008,47, 7079-7081

                                  144.Zhipeng Yu, Xiaohua Liu, Zhenhua Dong, Mingsheng Xie, Xiaoming Feng,* AnN,N′-Dioxide/In(OTf)3 Catalyst for the Asymmetric Hetero-Diels-Alder Reaction Between Danishefsky's Dienes and Aldehydes: Application in the Total Synthesis of Triketide,Angew. Chem., Int. Ed.2008,47, 1308-1311.

                                  145.Xin Zhou, Xiaohua Liu, Xu Yang, Deju Shang, Junguo Xin, Xiaoming Feng,* Highly Enantioselective Hydrophosphonylation of Aldehydes Catalyzed by Tridentate Schiff Base Aluminum(III) Complexes, Angew. Chem. Int. Ed.2008,47, 392-394.

                                  146.Yuehong Wen, Bo Gao, Yingzi Fu, Shunxi Dong, Xiaohua Liu, Xiaoming Feng,* Asymmetric Three-Component Strecker Reactions Catalyzed by trans-4-Hydroxy-L-proline-DerivedN,N′-Dioxides,Chem. Eur. J.2008,14, 6789-6795.

                                  147.Zongrui Hou, Jun Wang, Xiaohua Liu, Xiaoming Feng,* Highly Enantioselective Strecker Reaction of Ketoimines Catalyzed by an Organocatalyst from (S)-BINOL and L-Prolinamide,Chem. Eur. J.2008,14, 4484-4486.

                                  148.Jun Wang, Xiaolei Hu, Jun Jiang, Shaohua Gou, Xiao Huang, Xiaohua Liu, Xiaoming Feng,* Asymmetric Activation of tropos 2,2'-Biphenol with Cinchonine Generating a Remarkably Effective Catalyst for the Asymmetric Strecker Reaction of N-Ts Protected Aldimines and Ketoimines, Angew. Chem. Int. Ed.2007,46, 8468-8470.

                                  149.Yuehong Wen, Yan Xiong, Lu Chang, Jinglun Huang, Xiaohua Liu, Xiaoming Feng,* Chiral Bisformamides as Effective Organocatalysts for Asymmetric One-pot, Three-Component Strecker Reaction, J. Org. Chem.2007,72, 7715-7719.

                                  150.Xin Zhang, Donghui Chen, Xiaohua Liu, Xiaoming Feng,* Enantioselective Allylation of Ketones Catalyzed by N,N′-Dioxide and Indium(III) Complex, J. Org. Chem.2007,72, 5227-5233.

                                  151.Bo Qin, Xiaohua Liu., Jian Shi, Ke Zheng, Haitao Zhao, Xiaoming Feng,* Enantioselective Cyanosilylation of a,a-Dialkoxy Ketones Catalyzed by Proline-Derived in Situ Prepared N-Oxides as Bifunctional Organocatalysts, J. Org. Chem.2007,72, 2374-2378.

                                  152.Jinglun Huang, Xiaohua Liu, Yuehong Wen, Bo Qin, Xiaoming Feng,* Enantioselective Strecker Reaction of Phosphinoyl Ketoimines Catalyzed by in situ Prepared Chiral N,N′-Dioxides,J. Org. Chem.2007,72, 204-208.

                                  153.Xiao Huang, Jinglun Huang, Yuehong Wen, Xiaoming Feng,* Asymmetric Strecker Reaction of Ketoimines Catalyzed by a Novel Chiral Bifunctional N,N′-Dioxide,Adv. Synth. Catal.2006,348, 2579-2584.

                                  154.Yuehong Wen,Xiao Huang, Jinglun Huang, Yan Xiong, Bo Qin, Xiaoming Feng,* Asymmetric Cyanosilylation of Aldehydes Catalyzed by Novel Organocatalysts, Synlett2005, 2445-2448.

                                  155.Xiaohua Liu, Bo Qin, Bin He, Xiaoming Feng,* Catalytic Asymmetric Cyanosilylation of Ketones by a Chiral Amino Acid SaltJ. Am. Chem. Soc. 2005,127, 12224-12225.

                                  156.Fu-Xue Chen, Hui Zhou Xiaohua LiuBo Qin, Xiaoming Feng,*  Guolin Zhang, Yaozhong Jiang, Enantioselective Cyanosilylation Of Ketones by a Catalytic Double-Activation Method Using Aluminum Complex and N-oxide,Chem. Eur. J. 2004,10, 4790-4797.

                                  157.Xiaoming Feng, Lianhe Shu, Yian Shi*, Complete Conversion of Racemic Enol Ester Epoxides into Optically Active a-Acyloxy Ketones, J. Am. Chem. Soc.1999,121, 11002-11003.

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